SYNTHESIS OF THIAZOLE DERIVATIVES
Synthesis of Thiazole Derivatives and Evaluation of …
In this paper, we report the synthesis of TOTOBzl and TOTOEt together with the one- and two-dimensional 1H NMR investigations of complexes between these TOTO analogues and the dsDNA oligonucleotide d(CGCTAGCG)2.
Synthesis of Thiazole Derivatives—A Review - Pharma
Recently, heterocyclic compounds analogues and their derivatives have attracted strong interest in medicinal chemistry due to their biological and pharmacological properties. The small and simple benzothiazole nucleus possesses numerous biological properties like - antitumor, antimicrobial, anti-inflammatory, anticonvulsant, and antidiabetic activities. These activities are also possessed by its substituted derivatives as well. The present review focuses on some commonly used easy procedures to synthesize the benzothiazole moiety and its derivatives, which comprise of different biological activities.
Bachelor of Pharmacy - AIMST University
Devmurari et al., prepared a series of seven substituted 2-phenyl benzothiazoles and substituted 1, 3-benzothiazole-2-yl-4-carbothioate derivatives. All synthesized novel compounds were screened for anticancer activity and compounds (1.13) and (1.14) showed very good anticancer activity 35.
SYNTHESIS AND BIOLOGICAL EVALUATION OF …
Cheng K, Xue JY, Zhu HL. Design, synthesis and an- tibacterial activity studies o thiazole derivatives as po- tent eckAS inhibitors. Bioorg Med Chem Lett 2013;23:4235-4238.